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- 2005
Pharmacokinetic/pharmacodynamic modelling of the anti-hyperalgesic and anti-nociceptive effect of adenosine A1 receptor partial agonists in neuropathic pain,
Eur J Pharmacol, vol. 514, no. 2-3, pp. 131-40. DOI
Targeting liposomes with protein drugs to the blood-brain barrier in vitro,
Eur J Pharm Sci, vol. 25, no. 2-3, pp. 299-305. DOI
Brain penetration of synthetic adenosine A1 receptor agonists in situ: role of the rENT1 nucleoside transporter and binding to blood constituents,
Eur J Pharm Sci, vol. 24, no. 1, pp. 59-66. DOI
- 2004
Population pharmacokinetic-pharmacodynamic modelling of the anti-hyperalgesic effect of 5'deoxy-N6-cylopentyladenosine in the mononeuropathic rat,
Eur J Pharmacol, vol. 504, no. 1-2, pp. 7-15. DOI
Characterization and modulation of the transferrin receptor on brain capillary endothelial cells,
Pharm Res, vol. 21, no. 5, pp. 761-9.
Population pharmacokinetic modeling of blood-brain barrier transport of synthetic adenosine A1 receptor agonists,
J Pharmacol Exp Ther, vol. 311, no. 3, pp. 1138-46. DOI
Validation of the transferrin receptor for drug targeting to brain capillary endothelial cells in vitro,
J Drug Target, vol. 12, no. 3, pp. 145-50. DOI
Coupling of metal containing homing devices to liposomes via a maleimide linker: use of TCEP to stabilize thiol-groups without scavenging metals,
J Drug Target, vol. 12, no. 9-10, pp. 569-73. DOI
- 2003
Blood-brain barrier transport of synthetic adenosine A1 receptor agonists in vitro: structure transport relationships,
Eur J Pharm Sci, vol. 20, no. 3, pp. 347-56. DOI
Functional role of adenosine receptor subtypes in the regulation of blood-brain barrier permeability: possible implications for the design of synthetic adenosine derivatives,
Eur J Pharm Sci, vol. 19, no. 1, pp. 13-22. DOI
- 1997
Methodological considerations of intracerebral microdialysis in pharmacokinetic studies on drug transport across the blood-brain barrier,
Brain Res Brain Res Rev, vol. 25, no. 1, pp. 27-49. DOI
- 1995
Application of intracerebral microdialysis to study regional distribution kinetics of drugs in rat brain,
Br J Pharmacol, vol. 116, no. 5, pp. 2538-44.
The use of intracerebral microdialysis to determine changes in blood-brain barrier transport characteristics,
Pharm Res, vol. 12, no. 1, pp. 129-33.
Repeated microdialysis perfusions: periprobe tissue reactions and BBB permeability,
Brain Res, vol. 702, no. 1-2, pp. 261-5. DOI
The use of intracerebral microdialysis for the determination of pharmacokinetic profiles of anticancer drugs in tumor-bearing rat brain,
Pharm Res, vol. 12, no. 12, pp. 1924-31.
- 1994
Critical factors of intracerebral microdialysis as a technique to determine the pharmacokinetics of drugs in rat brain,
Brain Res, vol. 666, no. 1, pp. 1-8.
- 1993
Drug transport across the blood-brain barrier. III. Mechanisms and methods to improve drug delivery to the central nervous system,
Pharm World Sci, vol. 15, no. 1, pp. 2-9.
The use of intracerebral microdialysis to study blood-brain barrier transport in health, after modification and in disease,
Adv Exp Med Biol, vol. 331, pp. 257-62.
- 1992
Drug transport across the blood--brain barrier. I. Anatomical and physiological aspects,
Pharm Weekbl Sci, vol. 14, no. 5, pp. 305-10.
Drug transport across the blood-brain barrier. II. Experimental techniques to study drug transport,
Pharm Weekbl Sci, vol. 14, no. 6, pp. 338-48.
Modeling of the effect site equilibration kinetics and pharmacodynamics of racemic baclofen and its enantiomers using quantitative EEG effect measures,
J Pharmacol Exp Ther, vol. 261, no. 1, pp. 88-95.
Pharmacokinetic considerations on Orgaran (Org 10172) therapy,
Haemostasis, vol. 22, no. 2, pp. 73-84.
- 1991
Studies of interaction of a low-molecular-weight heparinoid (Org 10172) with cloxacillin and ticarcillin in healthy male volunteers,
Antimicrob Agents Chemother, vol. 35, no. 10, pp. 2110-5.
Influence of chlorthalidone on the pharmacokinetics and pharmacodynamics of Org 10172 (Lomoparan), a low molecular weight heparinoid, in healthy volunteers,
J Clin Pharmacol, vol. 31, no. 7, pp. 611-7.
The influence of Org 10172, a low molecular weight heparinoid, on antipyrine metabolism and the effect of enzyme induction on the response to Org 10172,
Br J Clin Pharmacol, vol. 32, no. 1, pp. 23-9.


